Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-7' and Ligand = 'BDBM50139124'
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of [125I] alpha bungarotoxin from rat alpha7 nACh receptor expressed in rat hippocampal membrane preincubated for 30 mins followed by ra...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
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Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataEC50: 6.00E+4nMAssay Description:Agonist activity at human alpha7 nACh receptor expressed in rat GH4C1 cells assessed as increase in current amplitudes after 2 to 3 days by patch cla...More data for this Ligand-Target Pair