Report error Found 3 Enz. Inhib. hit(s) with Target = 'Neurotensin receptor type 1' and Ligand = 'BDBM50257185'
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataIC50: 0.383nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Medical University of South Carolina
Curated by ChEMBL
Medical University of South Carolina
Curated by ChEMBL
Affinity DataEC50: 0.853nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
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