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Found 6 Enz. Inhib. hit(s) with Target = 'Neurotensin receptor type 1' and Ligand = 'BDBM50509510'
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 1 expressed in HT-29 cells incubated in dark after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 1 stably expressed in CHO cells incubated in dark after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human neurotensin receptor 1 in HT-29 cells assessed as intracellular calcium mobilization by Fura-2 dye based spectrofluorimetry...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataKd:  15nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 60 mins in presence of NT (8 to 13) without compound was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataKd:  3.60nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells preincubated for 20 mins to 2 hrs followed by addition of NT (8 to 13)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 75 mins in presence of NT (8 to 13) followed by compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed