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Found 3 Enz. Inhib. hit(s) with Target = 'Neurotensin receptor type 2' and Ligand = 'BDBM50019423'
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019423(CHEMBL3290105)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]NT at rat NTS2 overexpressed in CHOK1 cells after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019423(CHEMBL3290105)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as inhibition of SR142948a-induced calcium release by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50019423(CHEMBL3290105)
Affinity DataEC50:  19nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed