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Found 1 Enz. Inhib. hit(s) with Target = 'Nicotinamide N-methyltransferase' and Ligand = 'BDBM13016'
TargetNicotinamide N-methyltransferase(Homo sapiens (Human))
Utrecht University

LigandPNGBDBM13016(1,2,3,4-tetrahydroisoquinoline | CHEMBL14346 | THI...)
Affinity DataKi:  4.70E+7nM ΔG°:  -7.88kJ/molepH: 8.6 T: 2°CAssay Description:Enzyme activity assays were performed as previously described with NNMT (16.25 ug/mL, 550 nM) in 50 mM Tris buffer (pH 8.6) containing 1 mM DTT (all ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed