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Found 5 Enz. Inhib. hit(s) with Target = 'Nischarin' and Ligand = 'BDBM50050093'
TargetNischarin(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50050093((4-Chloro-6-methoxy-2-methyl-pyrimidin-5-yl)-imida...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]PIC from human imidazoline receptor 1 in human platelets analyzed under norepinephrine mask of alpha 2ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50050093((4-Chloro-6-methoxy-2-methyl-pyrimidin-5-yl)-imida...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-clonidine from bovine imidazoline receptor I-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50050093((4-Chloro-6-methoxy-2-methyl-pyrimidin-5-yl)-imida...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50050093((4-Chloro-6-methoxy-2-methyl-pyrimidin-5-yl)-imida...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50050093((4-Chloro-6-methoxy-2-methyl-pyrimidin-5-yl)-imida...)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed