Affinity DataKi: 0.830nMAssay Description:Binding affinity to human NOP receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.833nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at human NOP receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 31.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair