Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with Target = 'Nociceptin receptor' and Ligand = 'BDBM50210383'
TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50210383(4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol |...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I][14Tyr]nociceptin FQ from human cloned NOP receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50210383(4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol |...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I][14Tyr]nociceptin FQ from human cloned NOP receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50210383(4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol |...)
Affinity DataKi:  23nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50210383(4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol |...)
Affinity DataEC50:  331nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50210383(4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol |...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50210383(4-phenyl-1-(phenyl(o-tolyl)methyl)piperidin-4-ol |...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human NOP receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed