Found 4 Enz. Inhib. hit(s) with Target = 'Non-receptor tyrosine-protein kinase TNK1' and Ligand = 'BDBM2579'
TargetNon-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 0.584nMAssay Description:Inhibition of human TNK1 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human TNK1 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 2.5nMAssay Description:Binding constant for TNK1 kinase domainMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 2.5nMAssay Description:Binding constant for full-length TNK1More data for this Ligand-Target Pair