Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50203493'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Galderma R & D

Curated by ChEMBL
LigandPNGBDBM50203493(CHEMBL3912204)
Affinity DataIC50:  120nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Galderma R & D

Curated by ChEMBL
LigandPNGBDBM50203493(CHEMBL3912204)
Affinity DataIC50:  150nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL-17A release after 4 days by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed