Affinity DataIC50: 7nMAssay Description:Activity at biotinylated APC-labeled human RORgamma LBD assessed as of Induction of biotinylated SRC1 peptide recruitment incubated for 1 hr by TR-FR...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inverse agonist activity at GAL4-fused human RORgamma expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 18hr...More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) expressed in human Jurkat cells assessed as inhibition of IL-17F production after 20 hrs by luc...More data for this Ligand-Target Pair