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Found 4 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50203506'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50203506(CHEMBL3977048)
Affinity DataIC50:  7nMAssay Description:Activity at biotinylated APC-labeled human RORgamma LBD assessed as of Induction of biotinylated SRC1 peptide recruitment incubated for 1 hr by TR-FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50203506(CHEMBL3977048)
Affinity DataIC50:  17nMAssay Description:Inverse agonist activity at GAL4-fused human RORgamma expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 18hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50203506(CHEMBL3977048)
Affinity DataIC50:  44nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50203506(CHEMBL3977048)
Affinity DataIC50:  63nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) expressed in human Jurkat cells assessed as inhibition of IL-17F production after 20 hrs by luc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed