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Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50461086'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50461086(CHEMBL4228152)
Affinity DataIC50:  39nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) expressed in human HeLa-derived HG5LN cells transfected with the GAL4 DNA-binding domain fused ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed