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Found 3 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma [258-518]' and Ligand = 'BDBM221236'
TargetNuclear receptor ROR-gamma [258-518](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM221236(US9303015, 10a | US9303015, 10b | US9303015, 10c)
Affinity DataKd:  8.5nMpH: 7.0 T: 2°CAssay Description:ThermoFluor® experiments were carried out using instruments owned by Janssen Research and Discovery, L.L.C. through its acquisition of 3-Dimensio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [258-518](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM221236(US9303015, 10a | US9303015, 10b | US9303015, 10c)
Affinity DataKd:  39nMpH: 7.0 T: 2°CAssay Description:ThermoFluor® experiments were carried out using instruments owned by Janssen Research and Discovery, L.L.C. through its acquisition of 3-Dimensio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma [258-518](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM221236(US9303015, 10a | US9303015, 10b | US9303015, 10c)
Affinity DataKd:  3.40nMpH: 7.0 T: 2°CAssay Description:ThermoFluor® experiments were carried out using instruments owned by Janssen Research and Discovery, L.L.C. through its acquisition of 3-Dimensio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent