Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 2' and Ligand = 'BDBM50251070'
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50251070(CHEMBL464497 | N-(1-benzyl-1H-benzo[d]imidazol-5-y...)
Affinity DataEC50:  8.05nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50251070(CHEMBL464497 | N-(1-benzyl-1H-benzo[d]imidazol-5-y...)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed