Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Orexin/Hypocretin receptor type 1' and Ligand = 'BDBM50321514'
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50321514(((1S,5S)-6-(7-fluoroquinazolin-2-yl)-2,6-diazabicy...)
Affinity DataKi:  160nMAssay Description:Binding affinity to OX1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50321514(((1S,5S)-6-(7-fluoroquinazolin-2-yl)-2,6-diazabicy...)
Affinity DataIC50:  2.30E+3nMAssay Description:Antagonist activity at OX1R by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed