Affinity DataKi: 3.60nMAssay Description:Binding affinity to OX2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity to OX2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Binding affinity to OX2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Antagonist activity at OX2 receptor assessed as inhibition of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Antagonist activity at OX2 receptor assessed as inhibition of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Antagonist activity at OX2 receptor assessed as inhibition of calcium flux by FLIPR assayMore data for this Ligand-Target Pair