Affinity DataIC50: 23nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity P2X1 receptor in Apyrase pre-treated human platelets assessed as inhibition of collagen-induced platelet aggregation pre-incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMAssay Description:Antagonist activity P2X1 receptor in Apyrase pre-treated human platelets assessed as inhibition of TRAP6-induced platelet aggregation pre-incubated f...More data for this Ligand-Target Pair
Affinity DataIC50: 5.47E+3nMAssay Description:Antagonist activity P2X1 receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation pre-incubated for 30 mins before ADP ...More data for this Ligand-Target Pair