Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 4' and Ligand = 'BDBM50399207'
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  348nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx preincubated for 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  350nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced calcium flux measured for 30 secs at 0.4 s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at human P2X4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at human P2X4 receptor expressed in CHO cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at human P2X4 receptor expressed in CHO cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(RAT)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  750nMAssay Description:Antagonist activity at rat P2X4R expressed in HEK293 cells preincubated for 2 mins followed by ATP addition and measured after 4 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  3.71E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  3.99E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells by Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at P2X4R (unknown origin) expressed in 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by Fura-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by Fura-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  9.20E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Gwangju Institute of Science and Technology (GIST)

Curated by ChEMBL
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50:  9.20E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed