Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 7' and Ligand = 'BDBM50126724'
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126724(CHEMBL282808 | Isoquinoline-5-sulfonic acid 4-{(S)...)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126724(CHEMBL282808 | Isoquinoline-5-sulfonic acid 4-{(S)...)
Affinity DataIC50:  71nMAssay Description:Antagonistic activity against P2X7 receptor measured as the ATP dependent calcium influx in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed