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Found 2 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 1' and Ligand = 'BDBM50246518'
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246518(((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-d...)
Affinity DataKi:  100nMAssay Description:Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246518(((2R,3S,4S)-2-ethyl-3-methyl-4-(phenylamino)-3,4-d...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed