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Found 2 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 12' and Ligand = 'BDBM50445023'
TargetP2Y purinoceptor 12(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445023(CHEMBL3098234)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at P2Y12 receptor in rat platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445023(CHEMBL3098234)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at P2Y12 receptor in human platelet-rich plasma assessed as inhibition of ADP-induced platelet aggregation incubated for 5 mins p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed