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Found 3 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 14' and Ligand = 'BDBM50271102'
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50271102(((((2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin...)
Affinity DataIC50:  11nMAssay Description:Binding affinity to human P2Y14 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50271102(((((2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human recombinant P2Y14 receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation proximi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50271102(((((2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human P2Y14 receptor expressed in HEK293 cells coexpressing phospholipase C-activating Gi protein cells assessed as inhibition of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed