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Found 3 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 14' and Ligand = 'BDBM50343888'
TargetP2Y purinoceptor 14(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50343888((R)-4-(4-(2,2-difluoro-1-hydroxyethyl)phenyl)-7-(4...)
Affinity DataKi:  4nMAssay Description:Inhibition of mouse P2Y14 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50343888((R)-4-(4-(2,2-difluoro-1-hydroxyethyl)phenyl)-7-(4...)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of mouse P2Y14 receptor in presence of 2% HSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50343888((R)-4-(4-(2,2-difluoro-1-hydroxyethyl)phenyl)-7-(4...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at mouse P2Y14 receptor expressed in HEK293 cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed