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Found 1 Enz. Inhib. hit(s) with Target = 'PAS domain-containing serine/threonine-protein kinase' and Ligand = 'BDBM528478'
TargetPAS domain-containing serine/threonine-protein kinase(Homo sapiens (Human))
Bioenergenix

US Patent
LigandPNGBDBM528478(5-(2-Methoxyphenyl)-2-phenyl-[1,2,4]triazolo[1,5-a...)
Affinity DataIC50: <1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent