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Found 3 Enz. Inhib. hit(s) with Target = 'Palmitoleoyl-protein carboxylesterase NOTUM' and Ligand = 'BDBM50154391'
TargetPalmitoleoyl-protein carboxylesterase NOTUM(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50154391(CHEMBL3775257)
Affinity DataEC50:  88nMAssay Description:Inhibition of human notum pectinacetylesterase expressed in 293F cells after 30 mins by TCF/LEF cell sensor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPalmitoleoyl-protein carboxylesterase NOTUM(Homo sapiens (Human))
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50154391(CHEMBL3775257)
Affinity DataEC50:  88nMAssay Description:Inhibition of C-terminal His-V5 tagged human Notum expressed in human HEK293F cells harbouring TCF/LEF luciferase reporter gene assessed as activatio...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPalmitoleoyl-protein carboxylesterase NOTUM(Mus musculus)
Lexicon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50154391(CHEMBL3775257)
Affinity DataEC50:  342nMAssay Description:Inhibition of mouse notum pectinacetylesterase expressed in 293F cells after 30 mins by TCF/LEF cell sensor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed