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Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM33283'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM33283((3-{4-[(3-phenyl-7-propyl-1,2-benzisoxazol-6-yl)ox...)
Affinity DataKi:  0.300nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR gamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM33283((3-{4-[(3-phenyl-7-propyl-1,2-benzisoxazol-6-yl)ox...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at GAL4-tagged PPARdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM33283((3-{4-[(3-phenyl-7-propyl-1,2-benzisoxazol-6-yl)ox...)
Affinity DataEC50:  20nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR delta receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed