Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM50360740'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  3.00E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at GAL4-tagged PPARdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Canis familiaris)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at dog PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50: >4.20E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed