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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50267991'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50267991((R)-2-(3-(3-(4-methoxybenzoyl)-2-methyl-6-(trifluo...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H2]nTZD3 from human recombinant GST-fused PPARgamma expressed in Escherichia coli by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50267991((R)-2-(3-(3-(4-methoxybenzoyl)-2-methyl-6-(trifluo...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant PPARgamma expressed in COS1 cells coexpressing GAL4 assessed as transcriptional activity after 48 hrs by lucife...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed