Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50401011'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50401011(CHEMBL2206303)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to PPARgamma ligand binding domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50401011(CHEMBL2206303)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human GAL4-fused PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene transactivatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed