Found 4 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform' and Ligand = 'BDBM119531'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Curtin University
Curated by ChEMBL
Curtin University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Curtin University
Curated by ChEMBL
Curtin University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Curtin University
Curated by ChEMBL
Curtin University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF? Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufa...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Curtin University
Curated by ChEMBL
Curtin University
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF? Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufa...More data for this Ligand-Target Pair