Found 3 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform' and Ligand = 'BDBM50332019'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Affinity DataKd: 960nMAssay Description:Binding affinity to PI3Kalpha by high throughput assayMore data for this Ligand-Target Pair