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Found 4 Enz. Inhib. hit(s) with Target = 'Phosphoglycerate kinase 1' and Ligand = 'BDBM50216219'
TargetPhosphoglycerate kinase 1(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50216219(CHEMBL87680)
Affinity DataKd:  1.40E+5nMAssay Description:Dissociation constant for binding with Phosphoglycerate kinase (PGK) enzyme is evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoglycerate kinase 1(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50216219(CHEMBL87680)
Affinity DataKd:  1.19E+5nMAssay Description:Equilibrium binding affinity against histamine-167 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPhosphoglycerate kinase 1(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50216219(CHEMBL87680)
Affinity DataKd:  1.60E+5nMAssay Description:Equilibrium binding affinity against histamine-170 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPhosphoglycerate kinase 1(Homo sapiens (Human))
University Of Sheffield

Curated by ChEMBL
LigandPNGBDBM50216219(CHEMBL87680)
Affinity DataKd:  3.03E+5nMAssay Description:Equilibrium binding affinity against histamine-62 residue of phosphoglycerokinase in yeastMore data for this Ligand-Target Pair
In DepthDetails Article