Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Phosphopantetheine adenylyltransferase' and Ligand = 'BDBM82153'
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50:  8.80E+3nMAssay Description:The reverse assay was performed in polyproplene 96-well plates containing in each well either 1 uL DMSO, 1 UL of variable concentrations of test comp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Escherichia coli)
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50:  1.30E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphopantetheine adenylyltransferase(Enterococcus faecalis (Streptococcus faecalis))
Pfizer

LigandPNGBDBM82153(7-substituted pyrazoloquinolone, 12)
Affinity DataIC50: >6.50E+4nMAssay Description:PPAT screening assay (forward-direction assay) were performed in clear 384 well plates containing in each well either 1-uL DMSO, 1 uL of variable con...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed