Found 2 Enz. Inhib. hit(s) with Target = 'Pituitary adenylate cyclase-activating polypeptide type I receptor' and Ligand = 'BDBM50250079'
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataIC50: 8.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair