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Found 2 Enz. Inhib. hit(s) with Target = 'Plasma kallikrein' and Ligand = 'BDBM50431213'
TargetPlasma kallikrein(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl

Curated by ChEMBL
LigandPNGBDBM50431213(CHEMBL2332604)
Affinity DataKi:  0.300nMAssay Description:Inhibition of human recombinant polyhistidine-tagged plasma kallikrein expressed in Escherichia coli XL1 blue using Z-FR-AMC as substrate by fluorime...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl

Curated by ChEMBL
LigandPNGBDBM50431213(CHEMBL2332604)
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human PK using Z-Phe-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed