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Found 3 Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50005229'
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed