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Found 2 Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50011628'
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011628(4-(2-Chloro-phenyl)-2-iodo-9-methyl-6H-1-thia-5,7,...)
Affinity DataIC50:  370nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011628(4-(2-Chloro-phenyl)-2-iodo-9-methyl-6H-1-thia-5,7,...)
Affinity DataIC50:  370nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed