Found 8 Enz. Inhib. hit(s) with Target = 'Platelet-derived growth factor receptor alpha' and Ligand = 'BDBM50300690'
Affinity DataIC50: 42nMAssay Description:Inhibition of PDGFRalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human 3C cleavage site/N-terminal GST-His6 fused PDGFR alpha C-terminal fragment (Q551 to L1089 residues) harboring V561D m...More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to PDGFRAMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to PDGFRalpha (unknown origin) by KinomeSCan assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMAssay Description:Binding affinity to recombinant human PDGFRA (575 to 1002 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Binding affinity to PDGFRalphaMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to PDGFRalphaMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding constant for PDGFRA kinase domainMore data for this Ligand-Target Pair