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Found 2 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50130580'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50130580(3-Amino-5H-benzo[c][1,5]naphthyridin-6-one | 3-ami...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity against Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50130580(3-Amino-5H-benzo[c][1,5]naphthyridin-6-one | 3-ami...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant PARP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed