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Found 1 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily E/KQT member 1' and Ligand = 'BDBM50420056'
TargetPotassium voltage-gated channel subfamily E/KQT member 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420056(CHEMBL2046673)
Affinity DataIC50:  5.80E+3nMAssay Description:Antagonist activity at KCNQ1/MINK expressed in CHO cells assessed as inhibition of KCl-induced 86Rb+ efflux incubated for 10 mins prior to KCl-induct...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed