Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily H member 2' and Ligand = 'BDBM50095796'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50095796(CHEMBL3590496)
Affinity DataKi:  176nMAssay Description:Displacement of [3H]dofetilide from human Kv11.1 expressed in HEK293 cell membranes by competitive radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50095796(CHEMBL3590496)
Affinity DataKd:  125nMAssay Description:Binding affinity to human Kv11.1 expressed in HEK293 cell membranes assessed as binding affinity constant by [3H]dofetilide competition association a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed