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Found 10 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily H member 2' and Ligand = 'BDBM50117924'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory activity against Potassium channel HERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human ERG potassium channel in HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of human ERG current by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibitory concentration against potassium channel HERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibition of human Potassium channel HERG expressed in mammalian cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  7.76E+4nMAssay Description:Inhibition of human ERG in MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  7.76E+4nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv11.1 (ERG K+ channel) in open stateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117924(1-Cyclopropyl-6-fluoro-5-methyl-7-(3-methyl-pipera...)
Affinity DataIC50:  1.04E+5nMAssay Description:K+ channel blocking activity in Chinese hamster ovary cells expressing HERG Kv11.1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed