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Found 3 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50072708'
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072708(5-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-a...)
Affinity DataKi:  400nMAssay Description:Binding affinity was determined against hPR-A (human progesterone receptor) using progesterone radioligand in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072708(5-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-a...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity was determined against hPR (human progesterone receptor) compared to that of progesterone (100%)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072708(5-Methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-a...)
Affinity DataEC50:  75nMAssay Description:Antagonist activity against hPR (human progesterone receptor) compared to that of progesterone (100%)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed