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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50118698'
TargetProgesterone receptor(Homo sapiens (Human))
Women'S Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50118698(6-(3-Fluoro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo...)
Affinity DataIC50:  3.80nMAssay Description:Antagonist activity against progesterone receptor (PR) in an assay using PRE-luciferase plasmid co-transfected CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Women'S Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50118698(6-(3-Fluoro-phenyl)-4,4-dimethyl-1,4-dihydro-benzo...)
Affinity DataIC50:  8.20nMAssay Description:Antagonist activity against progesterone receptor (PR) in an alkaline phosphatase assay in the T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed