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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50355241'
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355241(CHEMBL1835834)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at human progesterone receptor in T47D cells after 24 hrs by alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355241(CHEMBL1835834)
Affinity DataIC50:  5.05E+4nMAssay Description:Displacement of [1,2,6,7-3H]PG from human PR-LBD after 24 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed