Found 4 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase FAP' and Ligand = 'BDBM50431242' TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of human FAP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School Of Biomedical Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human FAP using Z-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
