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Found 1 Enz. Inhib. hit(s) with Target = 'Protein O-GlcNAcase' and Ligand = 'BDBM139931'
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM139931(US8901087, 13)
Affinity DataKi:  0.400nM ΔG°:  -53.6kJ/molepH: 7.0 T: 2°CAssay Description:Enzymatic reactions are carried out in a reaction containing 50 mM NaH2PO4, 100 mM NaCl and 0.1% BSA (pH 7.0) using 2 mM 4-Methylumbelliferyl N-acety...More data for this Ligand-Target Pair
In DepthDetails US Patent