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Found 2 Enz. Inhib. hit(s) with Target = 'Protein arginine N-methyltransferase 1 [11-371]' and Ligand = 'BDBM50130929'
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of [3H]-U-69,593 binding to Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50130929(CHEMBL3633189)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4-derived peptide as substrate after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed