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Found 1 Enz. Inhib. hit(s) with Target = 'Protein c-Fos/Transcription factor Jun' and Ligand = 'BDBM50090444'
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090444(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50:  100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed