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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50048953'
LigandPNGBDBM50048953(4'-((R)-2-Amino-3-mercapto-propylamino)-biphenyl-3...)
Affinity DataIC50:  50nMAssay Description:Activity against rat brain FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50048953(4'-((R)-2-Amino-3-mercapto-propylamino)-biphenyl-3...)
Affinity DataIC50:  114nMAssay Description:In vitro inhibition of FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed